Publication Type
Peer Reviewed Journal
Mandatory Citation Fields
K. V. Rajendran, L. Kennedy, C. T. Oż Connor, E. Bergin and D. G. Gilheany
2013
Unknown
Tetrahedron Letters
Systematic survey of positive chlorine sources in the asymmetric Appel reaction: oxalyl chloride as a new phosphine activator
Published
Optional Fields
Please enter separate search keywords on separate lines
54
7009
7012

A wide selection of phosphine activators has been screened to improve the selection process in the asym- metric Appel reaction. Of the activators screened, hexachloroacetone (HCA) gave the highest selectivity with excellent yield, but at least one of its by-products, pentachloroacetone (PCA), can become involved in the selection process. In addressing this, a new reaction of phosphines with oxalyl chloride was discov- ered that can also generate the key intermediate chlorophosphonium salt (CPS), gives better enantiose- lectivity and possesses significant advantages over other phosphine activators. 

Grant Details
  • © University College Dublin 2010
  • Privacy
  • Policy
  • Freedom of Information